The database has 98685 Ki values for searching, and is growing. This list shows the Top 100 Receptors/Targets in Ki Please let us know if you feel we should add any papers or data. We welcome all feedback/suggestions/comments. Other features on Ki DB are: Download Ki, Data Mining, CDD Interface allows mining Ki database by structure, substructure or structure similarity. Anatomical profiling of GPCR expression is offered for selected targets.


Make a new search

Your search returned 165 results:

Download Data
IDReceptor/AliasesUniGeneAnat. ProfilingTest Ligand Name/AliasesNCIKi (nM)PubChemChEBIHot Ligand/AliasesSpeciesSourceReference
49995 5-HT Transporter  Aliases NCBI - UniGene N/A DOPAMINE  Aliases 173182 6,489.000000 PubChem-Compound ChEMBL 3H-5HT  Aliases RAT WHOLE BRAIN MINUS CEREBELLUM Rothman RB, et al., 2001
 
33037 5-HT Transporter  Aliases NCBI - UniGene N/A DOPAMINE  Aliases 173182 1,000.000000 PubChem-Compound ChEMBL 3H-GBR 12935  Aliases RAT BRAIN Andersen PH, et al., 1989
 
100415 5-HT Transporter  Aliases NCBI - UniGene N/A DOPAMINE  Aliases 173182 > 100,000.000000 PubChem-Compound ChEMBL 3H-IMIPRAMINE  Aliases HUMAN CLONED Tatsumi M, et al., 1997
 
15974 5-HT1A  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 545.000000 PubChem-Compound ChEMBL 125I-LSD  Aliases RAT CLONED Lovenberg TW, et al., 1993a
 
3347 5-HT1A  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 8,248.000000 PubChem-Compound ChEMBL 3H-8-OH-DPAT  Aliases HUMAN CLONED TOLL L, et. al., 1998
 
22265 5-HT1A  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 7,800.000000 PubChem-Compound ChEMBL 3H-8-OH-DPAT  Aliases RABBIT CEREBRAL CORTEX Weber JT, et al., 1997
 
20731 5-HT1A  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 > 10,000.000000 PubChem-Compound ChEMBL 3H-PAT  Aliases RAT HIPPOCAMPUS Gozlan H et al., 1983
 
20693 5-HT1A  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 > 10,000.000000 PubChem-Compound ChEMBL 3H-PAT  Aliases RAT STRIATUM Gozlan H et al., 1983
 
1027 5-HT1B  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 > 10,000.000000 PubChem-Compound ChEMBL 125I-CYP  Aliases RAT CORTEX MARKSTEIN ET AL, 1986
1031 5-HT1B  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 > 10,000.000000 PubChem-Compound ChEMBL 125I-CYP  Aliases RAT CORTEX HOYER, 1988(9) (J.R.R.)
 
1269 5-HT1D  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 > 10,000.000000 PubChem-Compound ChEMBL 3H-5HT  Aliases BOVINE STRIATUM HEURING & PEROUTKA, 1987
 
1910 5-HT2A  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 > 10,000.000000 PubChem-Compound ChEMBL 125I-LSD  Aliases HUMAN FR. CORTEX ELLIOT & KENT, 1989
 
1916 5-HT2A  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 > 10,000.000000 PubChem-Compound ChEMBL 125I-LSD  Aliases RAT CORTEX HARTIG ET AL., 1983
1919 5-HT2A  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 > 10,000.000000 PubChem-Compound ChEMBL 125I-LSD  Aliases RAT CORTEX KADAN ET AL., 1984
 
1915 5-HT2A  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 > 10,000.000000 PubChem-Compound ChEMBL 125I-LSD  Aliases BOVINE CAUDATE HARTIG ET AL., 1985
 
1920 5-HT2A  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 > 10,000.000000 PubChem-Compound ChEMBL 125I-MIL  Aliases RAT CORTEX HOFFMAN ET AL., 1987
 
1907 5-HT2A  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 > 10,000.000000 PubChem-Compound ChEMBL 3H-KETANSERIN  Aliases RAT CORTEX LYON ET AL., 1987
1912 5-HT2A  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 > 10,000.000000 PubChem-Compound ChEMBL 3H-KETANSERIN  Aliases RAT CORTEX MARKSTEIN ET AL, 1986
1914 5-HT2A  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 > 10,000.000000 PubChem-Compound ChEMBL 3H-KETANSERIN  Aliases RAT CORTEX HOYER, 1989 (J.R.R.)
 
3499 5-HT2A  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 > 10,000.000000 PubChem-Compound ChEMBL 3H-KETANSERIN  Aliases RAT CLONED TOLL L, et. al., 1998
 
1908 5-HT2A  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 > 10,000.000000 PubChem-Compound ChEMBL 3H-NMSP  Aliases RAT CORTEX LYON ET AL., 1986
 
1917 5-HT2A  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 > 10,000.000000 PubChem-Compound ChEMBL 3H-SPIPERONE  Aliases HUMAN CORTEX ANDORN ET AL., 1984
 
1909 5-HT2A  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 > 10,000.000000 PubChem-Compound ChEMBL 3H-SPIPERONE  Aliases RAT CORTEX LEYSEN ET AL., 1978
1918 5-HT2A  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 > 10,000.000000 PubChem-Compound ChEMBL 3H-SPIPERONE  Aliases RAT CORTEX CREESE & SNYDER, 1978
 
1911 5-HT2A  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 > 10,000.000000 PubChem-Compound ChEMBL 3H-SPIROPERIDOL  Aliases RAT CORTEX PEROUTKA & SNYDER, 1979
 
730 5-HT2C  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 > 10,000.000000 PubChem-Compound ChEMBL 125I-LSD  Aliases MOUSE C. PLEXUS TUM YAGALOFF ET AL., 1986
 
724 5-HT2C  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 > 10,000.000000 PubChem-Compound ChEMBL 125I-LSD  Aliases RAT Choroid Plexus YAMAMOTO & KEBABIAN, 1989
 
722 5-HT2C  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 6,030.000000 PubChem-Compound ChEMBL 125I-SCH 23982  Aliases PIG Choroid Plexus HOYER & KARPF, 1988
 
723 5-HT2C  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 > 10,000.000000 PubChem-Compound ChEMBL 125I-SCH 23982  Aliases RAT Choroid Plexus YAMAMOTO & KEBABIAN, 1989
 
725 5-HT2C  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 > 10,000.000000 PubChem-Compound ChEMBL 3H-MESULERGINE  Aliases PIG Choroid Plexus HOYER ET AL., 1986
727 5-HT2C  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 > 10,000.000000 PubChem-Compound ChEMBL 3H-MESULERGINE  Aliases PIG Choroid Plexus HOYER & KARPF, 1988
728 5-HT2C  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 > 10,000.000000 PubChem-Compound ChEMBL 3H-MESULERGINE  Aliases PIG Choroid Plexus HOYER, 1989 (J.R.R.)
729 5-HT2C  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 > 10,000.000000 PubChem-Compound ChEMBL 3H-MESULERGINE  Aliases PIG Choroid Plexus MARKSTEIN ET AL, 1986
 
3557 5-HT2C  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 > 10,000.000000 PubChem-Compound ChEMBL 3H-MESULERGINE  Aliases RAT CLONED TOLL L, et. al., 1998
3558 5-HT2C  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 > 10,000.000000 PubChem-Compound ChEMBL 3H-MESULERGINE  Aliases RAT CLONED TOLL L, et. al., 1998
 
2304 5-HT3  Aliases NCBI - UniGene N/A DOPAMINE  Aliases 173182 > 10,000.000000 PubChem-Compound ChEMBL 3H-BRL 43694  Aliases RAT CORTEX NELSON & THOMAS, 1989
 
3616 5-HT3  Aliases NCBI - UniGene N/A DOPAMINE  Aliases 173182 > 10,000.000000 PubChem-Compound ChEMBL 3H-GR-65630  Aliases MOUSE NG108-15 TOLL L, et. al., 1998
 
2307 5-HT3  Aliases NCBI - UniGene N/A DOPAMINE  Aliases 173182 > 10,000.000000 PubChem-Compound ChEMBL 3H-ZACOPRIDE  Aliases HUMAN HIPPOCAMPUS BARNES ET AL., 1989
 
2306 5-HT3  Aliases NCBI - UniGene N/A DOPAMINE  Aliases 173182 > 10,000.000000 PubChem-Compound ChEMBL 3H-ZACOPRIDE  Aliases HUMAN AMYGDALA BARNES ET AL., 1989
 
2303 5-HT3  Aliases NCBI - UniGene N/A DOPAMINE  Aliases 173182 > 10,000.000000 PubChem-Compound ChEMBL 3H-ZACOPRIDE  Aliases RAT ENTO CORTEX BARNES ET AL., 1988
 
16019 5-HT5  Aliases N/A N/A DOPAMINE  Aliases 173182 > 10,000.000000 PubChem-Compound ChEMBL 125I-LSD  Aliases MOUSE CLONED Plassat JL, et al., 1992
 
6435 5-HT5a  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 > 10,000.000000 PubChem-Compound ChEMBL 125I-LSD  Aliases MOUSE CLONED Matthes H, et.al., 1993
 
5229 5-HT5a  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 1,000.000000 PubChem-Compound ChEMBL 125I-LSD  Aliases RAT CLONED ERLANDER MG, ET AL., 1993
 
6448 5-HT5B  Aliases N/A N/A DOPAMINE  Aliases 173182 > 10,000.000000 PubChem-Compound ChEMBL 125I-LSD  Aliases MOUSE CLONED Matthes H, et.al., 1993
 
5230 5-HT5B  Aliases N/A N/A DOPAMINE  Aliases 173182 1,000.000000 PubChem-Compound ChEMBL 125I-LSD  Aliases RAT CLONED ERLANDER MG, ET AL., 1993
 
5226 5-HT5B  Aliases N/A N/A DOPAMINE  Aliases 173182 1,000.000000 PubChem-Compound ChEMBL 3H-5CT  Aliases RAT CLONED WISDEN W, ET AL., 1993
 
6612 5-HT6  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 > 10,000.000000 PubChem-Compound ChEMBL 3H-5HT  Aliases MOUSE CLONED PLASSAT JL, ET AL., 1993
 
15960 5-HT7  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 545.000000 PubChem-Compound ChEMBL 125I-LSD  Aliases RAT CLONED Lovenberg TW, et al., 1993a
 
6506 5-HT7  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 > 10,000.000000 PubChem-Compound ChEMBL 3H-5HT  Aliases HUMAN CLONED BARD JA, ET AL., 1993
 
5265 5-HT7  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 > 10,000.000000 PubChem-Compound ChEMBL 3H-5HT  Aliases RAT CLONED RUAT M, ET AL., 1993
35042 5-HT7  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 1,000.000000 PubChem-Compound ChEMBL 3H-5HT  Aliases RAT CLONED SHEN Y, ET AL., 1993
 
35041 5-HT7  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 1,000.000000 PubChem-Compound ChEMBL 3H-LSD  Aliases RAT CLONED SHEN Y, ET AL., 1993
 
20678 Adrenergic Alpha  Aliases N/A N/A DOPAMINE  Aliases 173182 250.000000 PubChem-Compound ChEMBL 3H-CLONIDINE  Aliases RAT BRAIN U'Prichard DC et al., 1977
29976 Adrenergic Alpha  Aliases N/A N/A DOPAMINE  Aliases 173182 240.000000 PubChem-Compound ChEMBL 3H-CLONIDINE  Aliases RAT BRAIN Greenberg, DA et al., 1976
Average245.00 
20596 Adrenergic Alpha  Aliases N/A N/A DOPAMINE  Aliases 173182 > 10,000.000000 PubChem-Compound ChEMBL 3H-WB4101  Aliases RAT BRAIN U'Prichard DC et al., 1977
30007 Adrenergic Alpha  Aliases N/A N/A DOPAMINE  Aliases 173182 > 10,000.000000 PubChem-Compound ChEMBL 3H-WB4101  Aliases RAT BRAIN Greenberg, DA et al., 1976
 
13171 adrenergic Alpha2  Aliases N/A N/A DOPAMINE  Aliases 173182 > 10,000.000000 PubChem-Compound ChEMBL 3H-IDAZOXAN  Aliases RAT BRAIN Boyajian CL, et al., 1987
 
12590 adrenergic Alpha2  Aliases N/A N/A DOPAMINE  Aliases 173182 9,989.000000 PubChem-Compound ChEMBL 3H-RAUWOLSCINE  Aliases RAT BRAIN Boyajian CL, et al., 1987
 
13297 adrenergic Beta  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 > 10,000.000000 PubChem-Compound ChEMBL 3H-DHA  Aliases Mammalian BRAIN Bylund DB, et al., 1976
 
50063 CANNABINOID CB1  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 1,000.000000 PubChem-Compound ChEMBL 3H-anandamide  Aliases theromyzon Tessulatum ganglia Stefano, GB et al., 1997
 
50064 CANNABINOID CB1  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 1,000.000000 PubChem-Compound ChEMBL 3H-anandamide  Aliases Hirudo medicinalis ganglia Stefano, GB et al., 1997
 
83261 D1  Aliases N/A N/A DOPAMINE  Aliases 173182 4,300.000000 PubChem-Compound ChEMBL 3H-SCH23390  Aliases HUMAN CLONED Janowsky A et al 2014
 
83278 D2  Aliases N/A N/A DOPAMINE  Aliases 173182 1,710.000000 PubChem-Compound ChEMBL 3H-YM 09151-2  Aliases HUMAN CLONED Janowsky A et al 2014
 
99698 D2  Aliases N/A N/A DOPAMINE  Aliases 173182 990.000000 PubChem-Compound ChEMBL [3H]spiperone  Aliases RAT CLONED Luo D et al 2016
 
83279 D3  Aliases N/A N/A DOPAMINE  Aliases 173182 61.000000 PubChem-Compound ChEMBL 3H-YM 09151-2  Aliases HUMAN CLONED Janowsky A et al 2014
 
99715 D3  Aliases N/A N/A DOPAMINE  Aliases 173182 101.000000 PubChem-Compound ChEMBL [3H]spiperone  Aliases RAT CLONED Luo D et al 2016
 
83280 D4  Aliases N/A N/A DOPAMINE  Aliases 173182 630.000000 PubChem-Compound ChEMBL 3H-YM 09151-2  Aliases HUMAN CLONED Janowsky A et al 2014
 
62933 DOPAMINE  Aliases N/A N/A DOPAMINE  Aliases 173182 22.000000 PubChem-Compound ChEMBL 3H-dopamine  Aliases CALF CAUDATE Creese, I et al., 1976a
 
62948 DOPAMINE  Aliases N/A N/A DOPAMINE  Aliases 173182 1,000.000000 PubChem-Compound ChEMBL 3H-Haloperidol  Aliases CALF CAUDATE Creese, I et al., 1976a
 
32871 DOPAMINE D1  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 130.000000 PubChem-Compound ChEMBL 125I-SCH 23982  Aliases HUMAN CLONED Michaelides MR, et al., 1995
 
20903 DOPAMINE D1  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 17.500000 PubChem-Compound ChEMBL 3H-dopamine  Aliases CALF BRAIN Burt DR et al., 1976
 
20874 DOPAMINE D1  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 16.800000 PubChem-Compound ChEMBL 3H-dopamine  Aliases CALF STRIATUM Burt DR et al., 1976
 
20924 DOPAMINE D1  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 11.700000 PubChem-Compound ChEMBL 3H-dopamine  Aliases CALF olfactory tubercle Burt DR et al., 1976
 
12531 DOPAMINE D1  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 > 10,000.000000 PubChem-Compound ChEMBL 3H-SCH23390  Aliases CANINE Choroid Plexus NICKLAUS ET AL., 1988
 
3196 DOPAMINE D1  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 4,470.000000 PubChem-Compound ChEMBL 3H-SCH23390  Aliases HUMAN CLONED TOLL L, et. al., 1998
16126 DOPAMINE D1  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 2,340.000000 PubChem-Compound ChEMBL 3H-SCH23390  Aliases HUMAN CLONED Sunahara RK, et al., 1991
Average3405.00 
67713 DOPAMINE D1  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 7,762.471166 PubChem-Compound ChEMBL 3H-SCH23390  Aliases PIG STRIATUM Gross, G. et, al. 1991
 
13122 DOPAMINE D1  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 1,450.000000 PubChem-Compound ChEMBL 3H-SCH23390  Aliases RAT STRIATUM Billard W, et al., 1984
16233 DOPAMINE D1  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 > 10,000.000000 PubChem-Compound ChEMBL 3H-SCH23390  Aliases RAT STRIATUM Neve KA, 1990
 
33864 DOPAMINE D1  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 380.000000 PubChem-Compound ChEMBL 3H-SCH23390  Aliases RAT FR. CORTEX Andersen PH, et al., 1985
 
15094 DOPAMINE D1  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 51.440000 PubChem-Compound ChEMBL 3H-SCH23390 High  Aliases BOVINE Pineal Simonneaux V., et. At., 1990
 
15098 DOPAMINE D1  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 > 10,000.000000 PubChem-Compound ChEMBL 3H-SCH23390 Low  Aliases BOVINE Pineal Simonneaux V., et. At., 1990
 
56240 DOPAMINE D1  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 124.000000 PubChem-Compound ChEMBL UNDEFINED  Aliases UNDEFINED UNDEFINED Herm L et al., 2009
 
16298 Dopamine D1A  Aliases N/A N/A DOPAMINE  Aliases 173182 > 10,000.000000 PubChem-Compound ChEMBL 125I-SCH 23982  Aliases HUMAN CLONED Tiberi M, et al., 1991
 
38618 Dopamine D1A  Aliases N/A N/A DOPAMINE  Aliases 173182 220.000000 PubChem-Compound ChEMBL Functional  Aliases RAT CLONED Qandil AM, et al., 2003
 
16312 Dopamine D1B  Aliases N/A N/A DOPAMINE  Aliases 173182 3,900.000000 PubChem-Compound ChEMBL 125I-SCH 23982  Aliases RAT CLONED Tiberi M, et al., 1991
 
64964 DOPAMINE D2  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 17.000000 PubChem-Compound ChEMBL 125I-7-OH-PIPAT  Aliases HAMSTER Ovary Hirose, Tsuyoshi. et. al, 2005
 
10825 DOPAMINE D2  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 710.000000 PubChem-Compound ChEMBL 125I-IODOSULPRIDE  Aliases HUMAN CLONED Freedman SB, et al., 1994
11677 DOPAMINE D2  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 544.000000 PubChem-Compound ChEMBL 125I-IODOSULPRIDE  Aliases HUMAN CLONED Sokoloff P, et al., 1992
13410 DOPAMINE D2  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 540.000000 PubChem-Compound ChEMBL 125I-IODOSULPRIDE  Aliases HUMAN CLONED Sautel F, et al., 1995
Average598.00 
16158 DOPAMINE D2  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 474.000000 PubChem-Compound ChEMBL 125I-IODOSULPRIDE  Aliases RAT CLONED Sokoloff P, et al., 1990
 
20907 DOPAMINE D2  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 670.000000 PubChem-Compound ChEMBL 3H-Haloperidol  Aliases CALF BRAIN Burt DR et al., 1976
 
20850 DOPAMINE D2  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 550.000000 PubChem-Compound ChEMBL 3H-Haloperidol  Aliases CALF STRIATUM Burt DR et al., 1976
 
14819 DOPAMINE D2  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 550.000000 PubChem-Compound ChEMBL 3H-Haloperidol  Aliases CALF Corpus Striatum Creese I, et al., 1976
 
14825 DOPAMINE D2  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 700.000000 PubChem-Compound ChEMBL 3H-Haloperidol  Aliases CALF olfactory tubercle Creese I, et al., 1976
20858 DOPAMINE D2  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 700.000000 PubChem-Compound ChEMBL 3H-Haloperidol  Aliases CALF olfactory tubercle Burt DR et al., 1976
Average700.00 
14831 DOPAMINE D2  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 475.000000 PubChem-Compound ChEMBL 3H-Haloperidol  Aliases CALF Nucleus accumbens Creese I, et al., 1976
20866 DOPAMINE D2  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 475.000000 PubChem-Compound ChEMBL 3H-Haloperidol  Aliases CALF Nucleus accumbens Burt DR et al., 1976
Average475.00 
12625 DOPAMINE D2  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 594.000000 PubChem-Compound ChEMBL 3H-Quinpirole  Aliases RAT BRAIN Levant B, et al., 1992
 
32988 DOPAMINE D2  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 > 10,000.000000 PubChem-Compound ChEMBL 3H-RACLOPRIDE  Aliases HUMAN CLONED Stormann TM, et al., 1990
 
13508 DOPAMINE D2  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 310.000000 PubChem-Compound ChEMBL 3H-S-Sulpiride  Aliases RAT STRIATUM Zahniser NR, et al., 1983
 
13520 DOPAMINE D2  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 250.000000 PubChem-Compound ChEMBL 3H-S-Sulpiride  Aliases RABBIT STRIATUM Zahniser NR, et al., 1983
 
32876 DOPAMINE D2  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 260.000000 PubChem-Compound ChEMBL 3H-SPIPERONE  Aliases HUMAN CLONED Michaelides MR, et al., 1995
 
16231 DOPAMINE D2  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 1,949.840000 PubChem-Compound ChEMBL 3H-SPIPERONE  Aliases MOUSE CLONED Neve KA, 1990
 
67721 DOPAMINE D2  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 2,187.761624 PubChem-Compound ChEMBL 3H-SPIPERONE  Aliases PIG STRIATUM Gross, G. et, al. 1991
 
12640 DOPAMINE D2  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 51.000000 PubChem-Compound ChEMBL 3H-SPIPERONE  Aliases RAT BRAIN Levant B, et al., 1992
 
13147 DOPAMINE D2  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 2,627.000000 PubChem-Compound ChEMBL 3H-SPIPERONE  Aliases RAT STRIATUM Billard W, et al., 1984
13530 DOPAMINE D2  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 210.000000 PubChem-Compound ChEMBL 3H-SPIPERONE  Aliases RAT STRIATUM Zahniser NR, et al., 1983
16234 DOPAMINE D2  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 8,912.500000 PubChem-Compound ChEMBL 3H-SPIPERONE  Aliases RAT STRIATUM Neve KA, 1990
Average3916.50 
33889 DOPAMINE D2  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 660.000000 PubChem-Compound ChEMBL 3H-SPIPERONE  Aliases RAT FR. CORTEX Andersen PH, et al., 1985
 
13543 DOPAMINE D2  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 200.000000 PubChem-Compound ChEMBL 3H-SPIPERONE  Aliases RABBIT STRIATUM Zahniser NR, et al., 1983
 
64971 DOPAMINE D2  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 576.000000 PubChem-Compound ChEMBL 3H-SPIPERONE  Aliases HAMSTER Ovary Hirose, Tsuyoshi. et. al, 2005
 
16056 DOPAMINE D2  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 211.000000 PubChem-Compound ChEMBL 3H-sulpiride  Aliases RAT Striatal Membranes Imafuku J, 1987
 
13380 DOPAMINE D2  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 20.000000 PubChem-Compound ChEMBL 3H-thymidine  Aliases HUMAN CLONED Sautel F, et al., 1995
 
3256 DOPAMINE D2  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 422.000000 PubChem-Compound ChEMBL 3H-YM 09151-2  Aliases HUMAN CLONED TOLL L, et. al., 1998
 
54782 DOPAMINE D2  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 450.000000 PubChem-Compound ChEMBL UNDEFINED  Aliases HUMAN UNDEFINED Dörfler M et al., 2008
54793 DOPAMINE D2  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 360.000000 PubChem-Compound ChEMBL UNDEFINED  Aliases HUMAN UNDEFINED Dörfler M et al., 2008
57070 DOPAMINE D2  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 2,100.000000 PubChem-Compound ChEMBL UNDEFINED  Aliases HUMAN UNDEFINED Pettersson F et al., 2010
57086 DOPAMINE D2  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 2.900000 PubChem-Compound ChEMBL UNDEFINED  Aliases HUMAN UNDEFINED Pettersson F et al., 2010
Average728.23 
32822 DOPAMINE D2 Long  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 7.500000 PubChem-Compound ChEMBL 3H-SPIPERONE  Aliases CANINE STRIATUM Van Tol, HH et al., 1991
 
37036 DOPAMINE D2 Long  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 1,606.000000 PubChem-Compound ChEMBL 3H-SPIPERONE  Aliases HUMAN CLONED Kilts JD, et al., 2002
 
32823 DOPAMINE D2 Long  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 2.800000 PubChem-Compound ChEMBL 3H-SPIPERONE  Aliases RAT CLONED Van Tol, HH et al., 1991
32824 DOPAMINE D2 Long  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 474.000000 PubChem-Compound ChEMBL 3H-SPIPERONE  Aliases RAT CLONED Van Tol, HH et al., 1991
Average238.40 
10834 DOPAMINE D3  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 29.000000 PubChem-Compound ChEMBL 125I-IODOSULPRIDE  Aliases HUMAN CLONED Freedman SB, et al., 1994
11699 DOPAMINE D3  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 23.000000 PubChem-Compound ChEMBL 125I-IODOSULPRIDE  Aliases HUMAN CLONED Sokoloff P, et al., 1992
13425 DOPAMINE D3  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 23.000000 PubChem-Compound ChEMBL 125I-IODOSULPRIDE  Aliases HUMAN CLONED Sautel F, et al., 1995
16984 DOPAMINE D3  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 54.950000 PubChem-Compound ChEMBL 125I-IODOSULPRIDE  Aliases HUMAN CLONED Cussac D, et al., 2000
Average32.49 
16182 DOPAMINE D3  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 25.000000 PubChem-Compound ChEMBL 125I-IODOSULPRIDE  Aliases RAT CLONED Sokoloff P, et al., 1990
 
12428 DOPAMINE D3  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 265.700000 PubChem-Compound ChEMBL 125I-NCQ 298  Aliases RAT CLONED Boundy VA, et al., 1993
 
66209 DOPAMINE D3  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 11.000000 PubChem-Compound ChEMBL 3H-7-OH-DPAT  Aliases RAT olfactory tubercle Campiani G, et al., 1998
 
16966 DOPAMINE D3  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 104.000000 PubChem-Compound ChEMBL 3H-S33084  Aliases HUMAN CLONED Cussac D, et al., 2000
 
16975 DOPAMINE D3  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 33.900000 PubChem-Compound ChEMBL 3H-SPIPERONE  Aliases HUMAN CLONED Cussac D, et al., 2000
 
13395 DOPAMINE D3  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 1.400000 PubChem-Compound ChEMBL 3H-thymidine  Aliases HUMAN CLONED Sautel F, et al., 1995
 
3311 DOPAMINE D3  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 20.000000 PubChem-Compound ChEMBL 3H-YM 09151-2  Aliases HUMAN CLONED TOLL L, et. al., 1998
 
54804 DOPAMINE D3  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 240.000000 PubChem-Compound ChEMBL UNDEFINED  Aliases HUMAN UNDEFINED Dörfler M et al., 2008
54827 DOPAMINE D3  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 72.000000 PubChem-Compound ChEMBL UNDEFINED  Aliases HUMAN UNDEFINED Dörfler M et al., 2008
Average156.00 
32859 DOPAMINE D4  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 28.000000 PubChem-Compound ChEMBL 3H-SPIPERONE  Aliases CANINE STRIATUM Van Tol, HH et al., 1991
 
54816 DOPAMINE D4  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 6.200000 PubChem-Compound ChEMBL UNDEFINED  Aliases HUMAN UNDEFINED Dörfler M et al., 2008
 
7053 DOPAMINE D4.2  Aliases N/A N/A DOPAMINE  Aliases 173182 180.000000 PubChem-Compound ChEMBL 3H-NGD 94-1  Aliases HUMAN CLONED TALLMAN JF, ET AL., 1997
 
7070 DOPAMINE D4.2  Aliases N/A N/A DOPAMINE  Aliases 173182 407.000000 PubChem-Compound ChEMBL 3H-YM 09151-2  Aliases HUMAN CLONED TALLMAN JF, ET AL., 1997
 
57984 DOPAMINE D4.4  Aliases N/A N/A DOPAMINE  Aliases 173182 100.600000 PubChem-Compound ChEMBL 35S-GTPGammaS  Aliases HUMAN CLONED Newman-Tancredi A, et al., 1997
 
13351 DOPAMINE D4.4  Aliases N/A N/A DOPAMINE  Aliases 173182 42.900000 PubChem-Compound ChEMBL 3H-SPIPERONE  Aliases HUMAN CLONED Newman-Tancredi A, et al., 1997
 
16153 DOPAMINE D5  Aliases NCBI - UniGene Anatomical Profiling DOPAMINE  Aliases 173182 228.000000 PubChem-Compound ChEMBL 3H-SCH23390  Aliases HUMAN CLONED Sunahara RK, et al., 1991
 
4617 Dopamine Transporter  Aliases NCBI - UniGene N/A DOPAMINE  Aliases 173182 1,770.000000 PubChem-Compound ChEMBL 3H-DA UPTAKE  Aliases HUMAN CLONED PRISTUPA ZB, ET AL., 1994
 
63565 Dopamine Transporter  Aliases NCBI - UniGene N/A DOPAMINE  Aliases 173182 1,700.000000 PubChem-Compound ChEMBL 3H-dopamine  Aliases RAT CLONED Wang W, et al., 2003
 
50019 Dopamine Transporter  Aliases NCBI - UniGene N/A DOPAMINE  Aliases 173182 38.300000 PubChem-Compound ChEMBL 3H-dopamine  Aliases RAT CAUDATE Rothman RB, et al., 2001
 
69510 Dopamine Transporter  Aliases NCBI - UniGene N/A DOPAMINE  Aliases 173182 66.000000 PubChem-Compound ChEMBL 3H-dopamine  Aliases RAT corpus striatum synaptosomes Richelson, E. et, al. 1984
 
4669 Dopamine Transporter  Aliases NCBI - UniGene N/A DOPAMINE  Aliases 173182 5,300.000000 PubChem-Compound ChEMBL 3H-GBR 12,935 BINDING  Aliases HUMAN CLONED PRISTUPA ZB, ET AL., 1994
 
33011 Dopamine Transporter  Aliases NCBI - UniGene N/A DOPAMINE  Aliases 173182 230.000000 PubChem-Compound ChEMBL 3H-GBR 12935  Aliases RAT STRIATUM Andersen PH, et al., 1989
 
100449 Dopamine Transporter  Aliases NCBI - UniGene N/A DOPAMINE  Aliases 173182 2,400.000000 PubChem-Compound ChEMBL 3H-WIN 35,428  Aliases HUMAN CLONED Tatsumi M, et al., 1997
 
63572 Dopamine Transporter  Aliases NCBI - UniGene N/A DOPAMINE  Aliases 173182 2,100.000000 PubChem-Compound ChEMBL 3H-WIN 35,428  Aliases RAT CLONED Wang W, et al., 2003
 
4652 Dopamine Transporter  Aliases NCBI - UniGene N/A DOPAMINE  Aliases 173182 5,900.000000 PubChem-Compound ChEMBL 3H-WIN 35,428 BINDING  Aliases HUMAN CLONED PRISTUPA ZB, ET AL., 1994
 
4635 Dopamine Transporter  Aliases NCBI - UniGene N/A DOPAMINE  Aliases 173182 67.000000 PubChem-Compound ChEMBL 3H-WIN 35,428 BINDING HIGH  Aliases HUMAN CLONED PRISTUPA ZB, ET AL., 1994
 
4659 Dopamine Transporter  Aliases NCBI - UniGene N/A DOPAMINE  Aliases 173182 3,100.000000 PubChem-Compound ChEMBL 3H-WIN 35,428 BINDING LOW  Aliases HUMAN CLONED PRISTUPA ZB, ET AL., 1994
 
38611 Dopamine1-like  Aliases N/A N/A DOPAMINE  Aliases 173182 1,000.000000 PubChem-Compound ChEMBL Functional  Aliases RAT STRIATUM Qandil AM, et al., 2003
 
17239 Dopamine2-like  Aliases N/A N/A DOPAMINE  Aliases 173182 880.000000 PubChem-Compound ChEMBL 3H-SCH23390  Aliases HUMAN STRIATUM Seeman P et al,1997b
 
17240 Dopamine2-like  Aliases N/A N/A DOPAMINE  Aliases 173182 192.000000 PubChem-Compound ChEMBL 3H-SCH23390  Aliases RAT STRIATUM Seeman P et al,1997b
 
33025 Norepinephrine transporter  Aliases N/A N/A DOPAMINE  Aliases 173182 1,000.000000 PubChem-Compound ChEMBL 3H-GBR 12935  Aliases RAT CEREBRAL CORTEX Andersen PH, et al., 1989
 
100431 Norepinephrine transporter  Aliases N/A N/A DOPAMINE  Aliases 173182 32,000.000000 PubChem-Compound ChEMBL 3H-Nisoxetine  Aliases HUMAN CLONED Tatsumi M, et al., 1997
 
10009 Norepinephrine transporter  Aliases N/A N/A DOPAMINE  Aliases 173182 323.000000 PubChem-Compound ChEMBL 3H-Norepinephrine  Aliases HUMAN CLONED Paczkowski,Bryan-Lluka,Porzgen,Bruss,Bonisch, 1999
 
10002 Norepinephrine transporter  Aliases N/A N/A DOPAMINE  Aliases 173182 392.000000 PubChem-Compound ChEMBL 3H-Norepinephrine  Aliases RAT CLONED Paczkowski,Bryan-Lluka,Porzgen,Bruss,Bonisch, 1999
 
49971 Norepinephrine transporter  Aliases N/A N/A DOPAMINE  Aliases 173182 40.300000 PubChem-Compound ChEMBL 3H-Norepinephrine  Aliases RAT WHOLE BRAIN MINUS CEREBELLUM Rothman RB, et al., 2001
 
10016 Norepinephrine transporter  Aliases N/A N/A DOPAMINE  Aliases 173182 397.000000 PubChem-Compound ChEMBL 3H-Norepinephrine  Aliases BOVINE CLONED Paczkowski,Bryan-Lluka,Porzgen,Bruss,Bonisch, 1999
 
47559 Sigma  Aliases N/A N/A DOPAMINE  Aliases 173182 > 10,000.000000 PubChem-Compound ChEMBL 3H-3-PPP,(+)  Aliases RAT BRAIN Largent BL, et al., 1984
 
16471 TA1  Aliases NCBI - UniGene N/A DOPAMINE  Aliases 173182 422.000000 PubChem-Compound ChEMBL 3H-Tyramine  Aliases HUMAN CLONED Borowsky B, et al.,2001